A New and Efficient Method for the Synthesis of Pyrimido[2,1-b]Benzothiazole Derivatives

نویسندگان

  • Fatemeh Chadegani
  • Fatemeh Darviche
  • Saeed Balalaie
چکیده

The one-pot three-component reaction of 2-aminobenzothiazole, benzaldehyde derivatives and β-ketoester, β-diketone or malonate derivatives in solvent-free conditions provides the corresponding pyrimido[2,1-b]benzothiazole derivatives at 60 ̊C in 60% 72% yields without using any catalyst in an optimistic time.

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تاریخ انتشار 2013